Life Chemicals is announcing the release of its G protein-coupled receptor kinase (GRK) Screening Set in a convenient assay-ready format. This collection includes 925 drug-like screening compounds with predicted inhibitory activity against GRKs (also known as GPCR kinases), selected from our proprietary HTS Compound Collection.
GRKs play a central role in regulating GPCR signaling, and their dysregulation has been implicated in cardiovascular diseases, neurological disorders, and metabolic syndromes. As such, they represent high-value targets in modern drug discovery.
- 10 mM solutions in DMSO
- volumes available: 10 µL, 25 µL, 50 µL, 100 µL
- 384-well microplates (Greiner bio-one ref: 781280 or 784201)
- Standard layout: 320 compounds per plate; columns 1-2 and 23-24 left empty
