Covalent Fragment Sets Freshly Pre-plated! Enjoy!

August 03, 2022

A newly created Pre-plated Covalent Fragment Screening Set is welcome to our vividly growing family of Pre-plated Fragment Screening Sets!

It includes 5,704 covalent inhibitor fragments, containing covalent warheads in assay-ready format, purchasable as one big screening set, or, alternatively, as four smaller complementary and non-overlapping subsets, selected to provide optimal structural diversity: 2.824, 1600, 960 and 320 and fragment-like covalent inhibitors.

Take advantage of conveniently concise and resourceful selections to boost your covalent screening and hit-finding FBDD projects!

This Pre-plated Covalent Fragment Screening Set is fully customizable, with variable concentrations and volumes provided in either 96- or 384-well plates.

Key features

  • Novel screening compounds synthesized in-house
  • Chemoinformatics assistance
  • Only drug-like molecules: Lipinski's Rule of Five and Veber criteria compliant
  • No PAINS (A, B, C families), toxic, reactive, and unstable compounds
  • Over 90 % purity confirmed by LCMS and/or NMR data
  • Hit re-supply, product scale-up
  • Compound library design, combinatorial synthesis based on hits found
  • Competitive pricing and convenient terms

Please, contact us at orders@lifechemicals.com for any additional information and price quotations.

For a detailed description and other formatting options, please, refer to the full Covalent Fragment Library.

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