Covalent Fragment Sets Freshly Pre-plated! Enjoy!

August 03, 2022

A newly created Pre-plated Covalent Fragment Screening Set is welcome to our vividly growing family of Pre-plated Fragment Screening Sets!

It includes 5,704 covalent inhibitor fragments, containing covalent warheads in assay-ready format, purchasable as one big screening set, or, alternatively, as four smaller complementary and non-overlapping subsets, selected to provide optimal structural diversity: 2,824, 1,600, 960 and 320 and fragment-like covalent inhibitors.

Take advantage of conveniently concise and resourceful selections to boost your covalent screening and hit-finding FBDD projects!

This Pre-plated Covalent Fragment Screening Set is fully customizable, with variable concentrations and volumes provided in either 96- or 384-well plates.

Key features

  • Novel screening compounds synthesized in-house
  • Chemoinformatics assistance
  • Only drug-like molecules: Lipinski's Rule of Five and Veber criteria compliant
  • No PAINS (A, B, C families), toxic, reactive, and unstable compounds
  • Over 90 % purity confirmed by LCMS and/or NMR data
  • Hit re-supply, product scale-up
  • Compound library design, combinatorial synthesis based on hits found
  • Competitive pricing and convenient terms

Please, contact us at for any additional information and price quotations.

For a detailed description and other formatting options, please, refer to the full Covalent Fragment Library.

Related products not to be missed:
This site uses cookies. Some of these cookies are essential, while others help us improve your experience by providing insights into how the site is being used. By using our website, you accept our conditions of use of cookies to track data and create content (including advertising) based on your interest. Accept