September 09, 2024
Our newest Pre-plated Covalent Inhibitor Screening Set is to become a perfect starting point for your covalent screening projects. Notably! This meticulously prepared selection of 4,800 structurally diverse covalent inhibitors contains a high variety of covalent warheads ready for immediate use!The screening compounds were picked out to possess optimal reactivity and essential stability, being compliant with our in-house MedChem and PAINS structural filters.
Please, contact us at orders@lifechemicals.com for any additional information and price quotations.
Even more covalent modifiers for cherry-picking and custom compound selection can be found in our Covalent Screening Library.
Please feel free to send your inquiries on a specific protein drug target needed, and our cheminformatics team will be happy to assist you in the structure optimization of potential irreversible binders, as well as in performing virtual covalent docking.
Make the most of our constantly-growing collection of readily available Pre-plated Screening Compound Sets for efficient hit finding in drug discovery projects.
Key features
- Novel screening compounds synthesized in-house
- Chemoinformatics assistance
- Only drug-like molecules, no PAINS, toxic, reactive, and unstable compounds
- Over 90 % purity confirmed by LCMS and/or NMR data
- Hit re-supply, product scale-up
- Compound library design and combinatorial synthesis based on found hits
- Competitive pricing and convenient terms